How Does Sildenafil Work?

The science behind Viagra explained simply. How PDE5 inhibitors improve blood flow.

Updated December 20255 min read

Simple Explanation

Sildenafil blocks an enzyme (PDE5) that normally restricts blood flow to the penis. With PDE5 blocked, blood vessels relax and expand, allowing more blood flow when you're aroused. It doesn't create arousal — it makes the physical response easier once you are aroused.

Step by Step

1. You Take Sildenafil

The medication absorbs into your bloodstream within 30-60 minutes.

2. PDE5 Enzyme Gets Blocked

Sildenafil inhibits PDE5, an enzyme that breaks down cGMP (a molecule that relaxes blood vessels).

3. cGMP Levels Rise

With PDE5 blocked, cGMP accumulates when you become aroused, causing smooth muscle relaxation.

4. Blood Flow Increases

Relaxed blood vessels allow more blood to flow into the penis, enabling a firmer erection.

Important: It's Not Automatic

Sildenafil doesn't cause spontaneous erections. You still need sexual stimulation and arousal. The medication just makes the physical response easier when arousal happens.

Think of it like clearing a blocked pipe — the water still needs to be turned on.

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